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DUSP6 – Hypogonadotropic Hypogonadism

Heterozygous variants in DUSP6 have been reported in patients with congenital hypogonadotropic hypogonadism (CHH), indicating an autosomal dominant inheritance pattern. In a sequencing study of 386 unrelated CHH individuals, five probands carried missense DUSP6 mutations, including c.566A>G (p.Asn189Ser) (PMID:23643382). A separate cohort of 196 Chinese patients identified four heterozygous DUSP6 variants in six affected individuals, without segregation to unaffected relatives (PMID:32389901). In total, 11 unrelated probands have been reported with DUSP6 variants, but no additional affected family members have been documented.

DUSP6 encodes the dual-specificity phosphatase MKP-3, a critical negative regulator of FGFR1–ERK signaling in GnRH neuron development. In vitro assays and interactome-based affiliation scoring support a role for DUSP6 loss in elevated ERK activity and defective GnRH secretion. Phosphorylation studies in cellular models demonstrate ERK1/2-mediated feedback on MKP-3 stability, underscoring mechanism relevance (PMID:15632084). Despite functional concordance, the paucity of segregation data and absence of CHH-specific animal models limit the evidence. Key take-home: DUSP6 variants likely contribute to CHH pathogenesis through ERK signaling dysregulation but require further familial and in vivo confirmation for diagnostic use.

References

  • American journal of human genetics • 2013 • Mutations in FGF17, IL17RD, DUSP6, SPRY4, and FLRT3 are identified in individuals with congenital hypogonadotropic hypogonadism. PMID:23643382
  • Journal of medical genetics • 2021 • Prevalence and associated phenotypes of DUSP6, IL17RD and SPRY4 variants in a large Chinese cohort with isolated hypogonadotropic hypogonadism. PMID:32389901
  • Molecular and cellular biology • 2005 • Extracellular signal-regulated kinases phosphorylate mitogen-activated protein kinase phosphatase 3/DUSP6 at serines 159 and 197, two sites critical for its proteasomal degradation. PMID:15632084

Evidence Based Scoring (AI generated)

Gene–Disease Association

Limited

11 probands across two cohorts; no segregation data; oligogenic modifiers noted

Genetic Evidence

Limited

11 unrelated CHH patients with heterozygous DUSP6 variants; lacking familial segregation

Functional Evidence

Moderate

In vitro and interactome analyses demonstrate DUSP6-ERK pathway dysregulation; feedback phosphorylation validated